Spallarossa, Andrea: шукати на сайті Z-Library

Рік:

2008

Мова:

english

Файл:

PDF, 383 KB

english, 2008

Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 1: Parallel synthesis, molecular modelling and structure–activity relationship studies on O-[2-(hetero)arylethyl]-N-phenylthiocarbamates

Sara Cesarini, Andrea Spallarossa, Angelo Ranise, Paola Fossa, Paolo La Colla, Giuseppina Sanna, Gabriella Collu, Roberta Loddo

Журнал:

Рік:

2008

Мова:

english

Файл:

PDF, 572 KB

english, 2008

Parallel one-pot synthesis and structure–activity relationship study of symmetric formimidoester disulfides as a novel class of potent non-nucleoside HIV-1 reverse transcriptase inhibitors

Sara Cesarini, Andrea Spallarossa, Angelo Ranise, Silvia Schenone, Olga Bruno, Paolo La Colla, Laura Casula, Gabriella Collu, Giuseppina Sanna, Roberta Loddo

Журнал:

Рік:

2008

Мова:

english

Файл:

PDF, 307 KB

english, 2008

6-Amino-4-oxo-1,3-diphenyl-2-thioxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl derivatives as a new class of potent inhibitors of Interleukin-8-induced neutrophil chemotaxis

Sara Cesarini, Andrea Spallarossa, Angelo Ranise, Olga Bruno, Nicoletta Arduino, Maria Bertolotto, Franco Dallegri, Massimiliano Tognolini, Thomas Gobbetti, Elisabetta Barocelli

Журнал:

Рік:

2009

Мова:

english

Файл:

PDF, 1.16 MB

english, 2009

Rational design, synthesis and biological evaluation of new 1,5-diarylpyrazole derivatives as CB1 receptor antagonists, structurally related to rimonabant

Giulia Menozzi, Paola Fossa, Elena Cichero, Andrea Spallarossa, Angelo Ranise, Luisa Mosti

Журнал:

Рік:

2008

Мова:

english

Файл:

PDF, 897 KB

english, 2008

N-Acylated and N,N′-diacylated imidazolidine-2-thione derivatives and N,N′-diacylated tetrahydropyrimidine-2(1H)-thione analogues: Synthesis and antiproliferative activity

Sara Cesarini, Andrea Spallarossa, Angelo Ranise, Silvia Schenone, Camillo Rosano, Paolo La Colla, Giuseppina Sanna, Bernardetta Busonera, Roberta Loddo

Журнал:

Рік:

2009

Мова:

english

Файл:

PDF, 424 KB

english, 2009

Novel modifications in the series of O-(2-phthalimidoethyl)-N-substituted thiocarbamates and their ring-opened congeners as non-nucleoside HIV-1 reverse transcriptase inhibitors

Andrea Spallarossa, Sara Cesarini, Angelo Ranise, Olga Bruno, Silvia Schenone, Paolo La Colla, Gabriella Collu, Giuseppina Sanna, Barbara Secci, Roberta Loddo

Журнал:

Рік:

2009

Мова:

english

Файл:

PDF, 580 KB

english, 2009

Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors: Docking-based CoMFA and CoMSIA analyses

Elena Cichero, Sara Cesarini, Paola Fossa, Andrea Spallarossa, Luisa Mosti

Журнал:

Рік:

2009

Мова:

english

Файл:

PDF, 2.51 MB

english, 2009

Parallel synthesis, molecular modelling and further structure–activity relationship studies of new acylthiocarbamates as potent non-nucleoside HIV-1 reverse transcriptase inhibitors

Andrea Spallarossa, Sara Cesarini, Angelo Ranise, Silvia Schenone, Olga Bruno, Alberto Borassi, Paolo La Colla, Margherita Pezzullo, Giuseppina Sanna, Gabriella Collu, Barbara Secci, Roberta Loddo

Журнал:

Medicinal Chemistry Research

Рік:

2009

Мова:

english

Файл:

PDF, 469 KB

english, 2009

(Hetero)aroyl esters of 2-(N-phthalimido)ethanol and analogues: parallel synthesis, anti-HIV-1 activity and cytotoxicity

Sara Cesarini, Andrea Spallarossa, Angelo Ranise, Silvia Schenone, Paolo La Colla, Gabriella Collu, Giuseppina Sanna, Roberta Loddo

Журнал:

Рік:

2010

Мова:

english

Файл:

PDF, 727 KB

english, 2010

Exploring the binding features of rimonabant analogues and acyclic CB1antagonists: docking studies and QSAR analysis

Elena Cichero, Giulia Menozzi, Andrea Spallarossa, Luisa Mosti, Paola Fossa

Журнал:

Journal of Molecular Modeling

Рік:

2008

Мова:

english

Файл:

PDF, 818 KB

english, 2008

Computational studies of the binding mode and 3D-QSAR analyses of symmetric formimidoester disulfides: a new class of non-nucleoside HIV-1 reverse transcriptase inhibitor

Elena Cichero, Sara Cesarini, Andrea Spallarossa, Luisa Mosti, Paola Fossa

Журнал:

Journal of Molecular Modeling

Рік:

2009

Мова:

english

Файл:

PDF, 513 KB

english, 2009

Acylthiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors: docking studies and ligand-based CoMFA and CoMSIA analyses

Elena Cichero, Sara Cesarini, Andrea Spallarossa, Luisa Mosti, Paola Fossa

Журнал:

Journal of Molecular Modeling

Рік:

2009

Мова:

english

Файл:

PDF, 529 KB

english, 2009

Synthesis and antiproliferative activity of basic thioanalogues of merbarone

Angelo Ranise, Andrea Spallarossa, Silvia Schenone, Olga Bruno, Francesco Bondavalli, Alessandra Pani, Maria Elena Marongiu, Valeria Mascia, Paolo La Colla, Roberta Loddo

Журнал:

Martino Bolognesi, Andrea Spallarossa, Paolo Ascenzi

Рік:

2003

Мова:

english

Файл:

PDF, 430 KB

english, 2003

Human rhinovirus 3C protease: a cysteine protease showing the trypsin(ogen)-like fold

Журнал:

Biochemistry and Molecular Biology Education

Рік:

2001

Мова:

english

Файл:

PDF, 400 KB

english, 2001

Homology modeling in tandem with 3D-QSAR analyses: A computational approach to depict the agonist binding site of the human CB2 receptor

Elena Cichero, Alessia Ligresti, Marco Allarà, Vincenzo di Marzo, Zelda Lazzati, Pasqualina D’Ursi, Anna Marabotti, Luciano Milanesi, Andrea Spallarossa, Angelo Ranise, Paola Fossa

Журнал:

Andrea Spallarossa, Janet L. Donahue, Timothy J. Larson, Martino Bolognesi, Domenico Bordo

Рік:

2011

Мова:

english

Файл:

PDF, 5.09 MB

english, 2011

Escherichia coli GlpE Is a Prototype Sulfurtransferase for the Single-Domain Rhodanese Homology Superfamily

Журнал:

Structure

Рік:

2001

Мова:

english

Файл:

PDF, 496 KB

english, 2001

The Three-Dimensional Structure of the Human NK Cell Receptor NKp44, a Triggering Partner in Natural Cytotoxicity

Claudia Cantoni, Marco Ponassi, Roberto Biassoni, Romana Conte, Andrea Spallarossa, Alessandro Moretta, Lorenzo Moretta, Martino Bolognesi, Domenico Bordo

Журнал:

Structure

Рік:

2003

Мова:

english

Файл:

PDF, 657 KB

english, 2003

Human rhinovirus 3C protease: a cysteine protease showing the trypsin(ogen)-like fold

Martino Bolognesi, Andrea Spallarossa, Paolo Ascenzi

Журнал:

Biochemistry and Molecular Biology Education

Рік:

2001

Мова:

english

Файл:

PDF, 242 KB

english, 2001

New Selective Phosphodiesterase 4D Inhibitors Differently Acting on Long, Short, and Supershort Isoforms

Bruno, Olga, Romussi, Alessia, Spallarossa, Andrea, Brullo, Chiara, Schenone, Silvia, Bondavalli, Francesco, Vanthuyne, Nicolas, Roussel, Christian

Журнал:

Biochemical and Biophysical Research Communications

Рік:

2009

Мова:

english

Файл:

PDF, 1.74 MB

english, 2009

Structure of the human NK cell triggering receptor NKp46 ectodomain

Marco Ponassi, Claudia Cantoni, Roberto Biassoni, Romana Conte, Andrea Spallarossa, Alessandra Pesce, Alessandro Moretta, Lorenzo Moretta, Martino Bolognesi, Domenico Bordo

Журнал:

Рік:

2003

Мова:

english

Файл:

PDF, 396 KB

english, 2003

Crystal structures of HIV-1 reverse transcriptase complexes with thiocarbamate non-nucleoside inhibitors

Andrea Spallarossa, Sara Cesarini, Angelo Ranise, Marco Ponassi, Torsten Unge, Martino Bolognesi

Журнал:

Biochemical and Biophysical Research Communications

Рік:

2008

Мова:

english

Файл:

PDF, 970 KB

english, 2008

The “Rhodanese” Fold and Catalytic Mechanism of 3-Mercaptopyruvate Sulfurtransferases: Crystal Structure of SseA from Escherichia coli

Andrea Spallarossa, Fabio Forlani, Aristodemo Carpen, Andrea Armirotti, Silvia Pagani, Martino Bolognesi, Domenico Bordo

Журнал:

Journal of Molecular Biology

Рік:

2004

Мова:

english

Файл:

PDF, 2.91 MB

english, 2004

Inhibition of Azotobacter vinelandii rhodanese by NO-donors

Andrea Spallarossa, Fabio Forlani, Silvia Pagani, Luca Salvati, Paolo Visca, Paolo Ascenzi, Martino Bolognesi, Domenico Bordo

Журнал:

Biochemical and Biophysical Research Communications

Рік:

2003

Мова:

english

Файл:

PDF, 176 KB

english, 2003

Anthrax toxin: a tripartite lethal combination

Paolo Ascenzi, Paolo Visca, Giuseppe Ippolito, Andrea Spallarossa, Martino Bolognesi, Cesare Montecucco

Журнал:

FEBS Letters

Рік:

2002

Мова:

english

Файл:

PDF, 228 KB

english, 2002

Identification of a Novel Pyrazolo[3,4- d ]pyrimidine Able To Inhibit Cell Proliferation of a Human Osteogenic Sarcoma in Vitro and in a Xenograft Model in Mice †

Manetti, Fabrizio, Santucci, Annalisa, Locatelli, Giada A., Maga, Giovanni, Spreafico, Adriano, Serchi, Tommaso, Orlandini, Maurizio, Bernardini, Giulia, Caradonna, Nicola P., Spallarossa, Andrea, Bru

Журнал:

Рік:

2007

Мова:

english

Файл:

PDF, 816 KB

english, 2007

Structure-Based Design, Parallel Synthesis, Structure−Activity Relationship, and Molecular Modeling Studies of Thiocarbamates, New Potent Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitor Isosteres of Phenethylthiazolylthiourea Derivatives

Ranise, Angelo, Spallarossa, Andrea, Cesarini, Sara, Bondavalli, Francesco, Schenone, Silvia, Bruno, Olga, Menozzi, Giulia, Fossa, Paola, Mosti, Luisa, La Colla, Massimiliano, Sanna, Giuseppina, Murre

Журнал:

Рік:

2005

Мова:

english

Файл:

PDF, 451 KB

english, 2005

Design, Synthesis, SAR, and Molecular Modeling Studies of Acylthiocarbamates: A Novel Series of Potent Non-nucleoside HIV-1 Reverse Transcriptase Inhibitors Structurally Related to Phenethylthiazolylthiourea Derivatives

Ranise, Angelo, Spallarossa, Andrea, Schenone, Silvia, Bruno, Olga, Bondavalli, Francesco, Vargiu, Laura, Marceddu, Tiziana, Mura, Massimo, La Colla, Paolo, Pani, Alessandra

Журнал:

Spallarossa, Andrea, Rotolo, Chiara, Sissi, Claudia, Marson, Giuseppe, Greco, Maria Laura, Ranise, Angelo, La Colla, Paolo, Busonera, Bernardetta, Loddo, Roberta

Рік:

2003

Мова:

english

Файл:

PDF, 227 KB

english, 2003

Further SAR studies on bicyclic basic merbarone analogues as potent antiproliferative agents

Журнал:

Ranise, Angelo, Lucchesini, Francesco, Caviglia, Matteo, Alfei, Silvana, Spallarossa, Andrea, Caneva, Chiara

Рік:

2013

Мова:

english

Файл:

PDF, 444 KB

english, 2013

Unconventional stereoselective one-pot synthesis of Knoevenagel-type indoles via in situ condensation of iminium salts with active methylene reagents

Журнал:

Tetrahedron

Рік:

2013

Мова:

english

Файл:

PDF, 838 KB

english, 2013

Enantio- and Diastereoselective Synthesis of Highly Substituted Benzazepines by a Multicomponent Strategy Coupled with Organocatalytic and Enzymatic Procedures

Moni, Lisa, Banfi, Luca, Basso, Andrea, Galatini, Andrea, Spallarossa, Martina, Riva, Renata

Журнал:

Journal of Organic Chemistry

Рік:

2014

Мова:

english

Файл:

PDF, 883 KB

english, 2014

Synthesis and biological evaluation of (acyl)hydrazones and thiosemicarbazones obtained via in situ condensation of iminium salts with nitrogen-containing nucleophiles

Caneva, Chiara, Alfei, Silvana, De Maria, Monica, Ibba, Cristina, Delogu, Ilenia, Spallarossa, Andrea, Loddo, Roberta

Журнал:

Molecular Diversity

Рік:

2015

Мова:

english

Файл:

PDF, 1.36 MB

english, 2015

Unconventional Knoevenagel-type Indoles: Synthesis and Cell-based Studies for the Identification of Pro-apoptotic Agents

Spallarossa, Andrea, Caneva, Chiara, Caviglia, Matteo, Alfei, Silvana, Butini, Stefania, Campiani, Giuseppe, Gemma, Sandra, Brindisi, Margherita, Zisterer, Daniela M., Bright, Sandra A., Williams, Cli

Журнал:

Ascenzi, Paolo, Bocedi, Alessio, Bolognesi, Martino, Spallarossa, Andrea, Coletta, Massimo, Cristofaro, Raimondo, Menegatti, Enea

Рік:

2015

Мова:

english

Файл:

PDF, 1.42 MB

english, 2015

Unprecedented One-Pot Stereoselective Synthesis of Knoevenagel-Type Derivatives via in situ Condensation of N -Methyleniminium Salts of Ethylenethiourea and Ethyleneurea with Active Methylene Reagents

Ranise, Angelo, Cesarini, Sara, Spallarossa, Andrea, Sancassan, Fernando, Bondavalli, Francesco, Bruno, Olga, Schenone, Silvia, Menozzi, Giulia, Fossa, Paola, Mosti, Luisa

Журнал:

Synthesis

Рік:

2007

Мова:

english

Файл:

PDF, 145 KB

english, 2007

The Bovine Basic Pancreatic Trypsin Inhibitor (Kunitz Inhibitor): A Milestone Protein

Журнал:

Current Protein & Peptide Science

Рік:

2003

Мова:

english

Файл:

PDF, 297 KB

Zoppi, Vittoria, Hughes, Scott J, Maniaci, Chiara, TESTA, ANDREA, Gmaschitz, Teresa, Wieshofer, Corinna, Koegl, Manfred, Riching, Kristin, Daniels, Danette L., Spallarossa, Andrea, Ciulli, Alessio

Журнал: